SAR study of 5-alkynyl substituted quinazolin-4(3H)-ones as phosphoinositide 3-kinase delta (PI3Kδ) inhibitors

Author:

Wei Manman,Zhang Xi,Wang Xiang,Song Zilan,Ding Jian,Meng Ling-Hua,Zhang AoORCID

Funder

National Natural Science Foundation of China

Shanghai Commission of Science and Technology

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference35 articles.

1. The phosphoinositide 3-kinase pathway;Cantley;Science,2002

2. Phosphoinositide 3-kinases: a conserved family of signal transducers;Vanhaesebroeck;Trends Biochem. Sci.,1997

3. The emerging mechanisms of isoform-specific PI3K signaling;Vanhaesebroeck;Nat. Rev. Mol. Cell Biol.,2010

4. Phosphatidylinositol 3-kinase inhibitors: promising drug candidates for cancer therapy;Kong;Cancer Sci.,2008

5. p110δ, a novel phosphatidylinositol 3-kinase catalytic subunit that associates with p85 and is expressed predominantly in leukocytes;Chantry;J. Biol. Chem.,1997

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