Fused heterocycles bearing bridgehead nitrogen as potent HIV-1 NNRTIs. Part 4: Design, synthesis and biological evaluation of novel imidazo[1,2-a]pyrazines-Reference-Cited by-同舟云学术

Fused heterocycles bearing bridgehead nitrogen as potent HIV-1 NNRTIs. Part 4: Design, synthesis and biological evaluation of novel imidazo[1,2-a]pyrazines

Published:2015-03 Issue: Volume:93 Page:330-337
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Huang Boshi,Liang Xin,Li Cuicui,Chen Wenmin,Liu Tao,Li Xiao,Sun Yueyue,Fu Lu,Liu Huiqing,De Clercq Erik,Pannecouque Christophe,Zhan Peng,Liu Xinyong

Funder

Key Project of National Natural Science Foundation of China

National Natural Science Foundation of China

Research Fund for the Doctoral Program of Higher Education of China

Natural Science Foundation of Shandong Province

KU Leuven

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference21 articles.

1. UNAIDS Gap Report,2014

2. HIV-1 NNRTIs: structural diversity, pharmacophore similarity, and implications for drug design;Zhan;Med. Res. Rev.,2013

3. Design strategies of novel NNRTIs to overcome drug resistance;Zhan;Curr. Med. Chem.,2009

4. Strategies for the design of HIV-1 non-nucleoside reverse transcriptase inhibitors: lessons from the development of seven representative paradigms;Li;J. Med. Chem.,2012

5. Recent advances in DAPYs and related analogues as HIV-1 NNRTIs;Chen;Curr. Med. Chem.,2011

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