Discovery of novel piperidine-substituted indolylarylsulfones as potent HIV NNRTIs via structure-guided scaffold morphing and fragment rearrangement-Reference-Cited by-同舟云学术

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Discovery of novel piperidine-substituted indolylarylsulfones as potent HIV NNRTIs via structure-guided scaffold morphing and fragment rearrangement

Published:2017-01 Issue: Volume:126 Page:190-201
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Li Xiao,Gao Ping,Huang Boshi,Zhou Zhongxia,Yu Zhao,Yuan Zheng,Liu Huiqing,Pannecouque Christophe,Daelemans Dirk,De Clercq Erik,Zhan Peng,Liu Xinyong

Funder

National Natural Science Foundation of China

Key Project of NSFC for International Cooperation

Natural Science Foundation of Shandong Province

Young Scholars Program of Shandong University

Major Project of Science and Technology of Shandong Province

KU Leuven

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference55 articles.

1. The first postmodern pandemic: 25 years of HIV/AIDS;Kallings;J. Intern. Med.,2008

2. Global Report: UNAIDS Report on the Global AIDS Epidemic,2015

3. Anti-HIV drugs: 25 compounds approved within 25 years after the discovery of HIV;De Clercq;Int. J. Antimicrob. Agents,2009

4. Twenty-six years of anti-HIV drug discovery: where do we stand and where do we go?;Mehellou;J. Med. Chem.,2010

5. Combined approaches for HIV cure;Margolis;Curr. Opin. HIV AIDS,2013

Cited by 20 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Deciphering the enigmas of non‐nucleoside reverse transcriptase inhibitors (NNRTIs): A medicinal chemistry expedition towards combating HIV drug resistance;Medicinal Research Reviews;2024-08-26

2. Structure‐based design, synthesis, and biological characterization of indolylarylsulfone derivatives as novel human immunodeficiency virus type 1 inhibitors with potent antiviral activities and favorable drug‐like profiles;Journal of Medical Virology;2024-07-29

3. Discovery of novel sulfonamide substituted indolylarylsulfones as potent HIV-1 inhibitors with better safety profiles;Acta Pharmaceutica Sinica B;2023-06

4. Chemical space exploration around indolylarylsulfone scaffold led to a novel class of highly active HIV-1 NNRTIs with spiro structural features;European Journal of Medicinal Chemistry;2022-08

5. An Overview on Indole Aryl Sulfide/Sulfone (IAS) as Anti‐HIV Non‐Nucleoside Reverse Transcriptase Inhibitors (NNRTIs);Asian Journal of Organic Chemistry;2022-02-19

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