Chemical space exploration around indolylarylsulfone scaffold led to a novel class of highly active HIV-1 NNRTIs with spiro structural features-Reference-Cited by-同舟云学术

Chemical space exploration around indolylarylsulfone scaffold led to a novel class of highly active HIV-1 NNRTIs with spiro structural features

Published:2022-08 Issue: Volume:238 Page:114471
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Gao Shenghua,Cheng Yusen,Song Shu,Song Letian,Zhao Fabao,Xu Shujing,Kang Dongwei,Sun Lin,Gao Ping,De Clercq Erik,Pannecouque Christophe,Liu Xinyong,Zhan Peng^ORCID

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference36 articles.

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2. Recent advances in the development of integrase inhibitors for HIV treatment;Trivedi;Curr. HIV AIDS Rep.,2020

3. HIV-1 fusion inhibitors targeting the membrane-proximal external region of Env spikes;Xiao;Nat. Chem. Biol.,2020

4. Retroviral DNA integration;Lesbats;Chem. Rev.,2016

5. The journey of HIV-1 non-nucleoside reverse transcriptase inhibitors (NNRTIs) from lab to clinic;Namasivayam;J. Med. Chem.,2019

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1. Deciphering the enigmas of non‐nucleoside reverse transcriptase inhibitors (NNRTIs): A medicinal chemistry expedition towards combating HIV drug resistance;Medicinal Research Reviews;2024-08-26

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3. Identification of Ebselen derivatives as novel SARS-CoV-2 main protease inhibitors: Design, synthesis, biological evaluation, and structure-activity relationships exploration;Bioorganic & Medicinal Chemistry;2023-12

4. Quinolines and isoquinolines as HIV-1 inhibitors: Chemical structures, action targets, and biological activities;Bioorganic Chemistry;2023-07

5. Discovery of novel sulfonamide substituted indolylarylsulfones as potent HIV-1 inhibitors with better safety profiles;Acta Pharmaceutica Sinica B;2023-06