Synthesis, computational and experimental pharmacological studies for (thio)ether-triazine 5-HT6R ligands with noticeable action on AChE/BChE and chalcogen-dependent intrinsic activity in search for new class of drugs against Alzheimer's disease-Reference-Cited by-同舟云学术

Synthesis, computational and experimental pharmacological studies for (thio)ether-triazine 5-HT6R ligands with noticeable action on AChE/BChE and chalcogen-dependent intrinsic activity in search for new class of drugs against Alzheimer's disease

Published:2023-11 Issue: Volume:259 Page:115695
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Czarnota-Łydka Kinga,Sudoł-Tałaj Sylwia,Kucwaj-Brysz Katarzyna,Kurczab Rafał,Satała Grzegorz,de Candia Modesto,Samarelli Francesco,Altomare Cosimo Damiano,Carocci Alessia,Barbarossa Alexia,Żesławska Ewa,Głuch-Lutwin Monika,Mordyl Barbara,Kubacka Monika,Wilczyńska-Zawal Natalia,Jastrzębska-Więsek Magdalena,Partyka Anna,Khan Nadia,Więcek Małgorzata,Nitek Wojciech,Honkisz-Orzechowska Ewelina,Latacz Gniewomir,Wesołowska Anna,Carrieri Antonio,Handzlik Jadwiga^ORCID

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference111 articles.

1. Review on Alzheimer's disease: inhibition of amyloid beta and tau tangle formation;Ashrafian;Int. J. Biol. Macromol.,2021

2. Molecular pathogenesis of alzheimer's disease: an update;Sanabria-Castro;Ann. Neurosci.,2017

3. Synaptic degeneration in Alzheimer disease;Makis;Nat. Rev. Neurol.,2022

4. A mechanistic survey of Alzheimer's disease;Tang;Biophys. Chem.,2022

5. Cholinesterase inhibitors as Alzheimer’s therapeutics (Review);Sharma;Mol. Med. Rep.,2019

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