4-Phenylureido/thioureido-substituted 2,2-dimethylchroman analogs of cromakalim bearing a bulky ‘carbamate’ moiety at the 6-position as potent inhibitors of glucose-sensitive insulin secretion-Reference-Cited by-同舟云学术

4-Phenylureido/thioureido-substituted 2,2-dimethylchroman analogs of cromakalim bearing a bulky ‘carbamate’ moiety at the 6-position as potent inhibitors of glucose-sensitive insulin secretion

Published:2016-10 Issue: Volume:121 Page:338-351
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Pirotte Bernard,Florence Xavier,Goffin Eric,Medeiros Marlen Borges,de Tullio Pascal,Lebrun Philippe

Funder

National Fund for Scientific Research

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

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4. Intracellular ATP directly blocks K+ channels in pancreatic B-cells;Cook;Nature,1984

5. ATP-sensitive potassium channels: structures, functions, and pathophysiology;Inagaki;Jpn. J. Physiol.,1998

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