Automated high-throughput in vitro assays to identify metabolic hotspots and protease stability of structurally diverse, pharmacologically active peptides for inhalation-Reference-Cited by-同舟云学术

Automated high-throughput in vitro assays to identify metabolic hotspots and protease stability of structurally diverse, pharmacologically active peptides for inhalation

Published:2022-03 Issue: Volume:211 Page:114518
ISSN:0731-7085
Container-title:Journal of Pharmaceutical and Biomedical Analysis
language:en
Short-container-title:Journal of Pharmaceutical and Biomedical Analysis

Author:

Wesche Frank,De Maria Leonardo,Leek Tomas,Narjes Frank,Bird James,Su Wu,Czechtizky Werngard

Publisher

Elsevier BV

Subject

Clinical Biochemistry,Spectroscopy,Drug Discovery,Pharmaceutical Science,Analytical Chemistry

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4. New modalities for challenging targets in drug discovery;Valeur;Angew. Chem. Int. Ed.,2017

5. Synthesis and incorporation into cyclic peptides of tolan amino acids and their hydrogenated congeners: construction of an array of A–B-loop mimetics of the Cε3 domain of human IgE;Offermann;J. Org. Chem.,2012

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