Fatty acid acylated peptide therapeutics: discovery of omega-n oxidation of the lipid chain as a novel metabolic pathway in preclinical species

Author:

Esposito SimoneORCID,Krick Alain,Pasquier Olivier,Bonche Fabrice,Ingenito Raffaele,Magotti Paola,Bianchi Elisabetta,Monteagudo Edith,Gallo Mariana,Cicero Daniel Oscar,Orsatti Laura,Veneziano Maria,Caretti Fulvia,Mele Riccardo,Roversi Daniela,Gennari Nadia,Brasseur Denis,Gauzy-Lazo Laurence,Duclos Olivier,Mauriac Christine,Illiano Stephane,Mallart Sergio

Publisher

Elsevier BV

Subject

Clinical Biochemistry,Spectroscopy,Drug Discovery,Pharmaceutical Science,Analytical Chemistry

Reference33 articles.

1. Peptide-based Drug Discovery,2017

2. Peptide therapeutics: current status and future directions;Fosgerau;Drug Discov. Today,2015

3. The current state of peptide drug discovery: back to the future;Henninot;? J. Med. Chem.,2018

4. Therapeutic peptides: historical perspectives, current development trends, and future directions;Lau;Bioorg. Med. Chem.,2018

5. Trends in peptide drug discovery;Muttenthaler;Nat. Rev. Drug Discov.,2021

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