In vitroand in vivo investigation of metabolic fate of riociguat by HPLC-Q-TOF/MS/MS and in silico evaluation of the metabolites by ADMET predictor™

Author:

Tiwari Shristy S.,Chavan Balasaheb B.,Kushwah Bhoopendra S.,Yerra Naga Veera,Mukesh Sumit,Sangamwar Abhay T.,Thaota Jagadeshwar Reddy,Talluri M.V.N. Kumar

Publisher

Elsevier BV

Subject

Clinical Biochemistry,Spectroscopy,Drug Discovery,Pharmaceutical Science,Analytical Chemistry

Reference33 articles.

1. Cellular and molecular pathobiology of pulmonary arterial hypertension;Humbert;J. Am. Coll. Cardiol.,2004

2. Cellular and molecular basis of pulmonary arterial hypertension;Morrell;J. Am. Coll. Cardiol.,2009

3. Riociguat for the treatment of pulmonary hypertension;Hambly;Expert Rev. Respir. Med.,2015

4. https://www.accessdata.fda.gov/drugsatfda_docs/label/2017/204819s006lbl.pdf, (Accessed 1 January 2018).

5. http://www.ema.europa.eu/docs/en_GB/document_library/EPAR_Public_assessment_report/human/002737/WC500165036.pdf, (Accessed 1 January 2017).

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