Synthesis and cross coupling of a highly substituted 2-pyridylboronate: application to the large scale synthesis of a mineralocorticoid antagonist-Reference-Cited by-同舟云学术

Synthesis and cross coupling of a highly substituted 2-pyridylboronate: application to the large scale synthesis of a mineralocorticoid antagonist

Published:2011-12 Issue:52 Volume:52 Page:7025-7029
ISSN:0040-4039
Container-title:Tetrahedron Letters
language:en
Short-container-title:Tetrahedron Letters

Author:

Boos Charles,Bowles Daniel M.,Cai Cuiman,Casimiro-Garcia Agustin,Chen Xiangyang,Hulford Catherine A.,Jennings Sandra M.,Jason Kiser E.,Piotrowski David W.,Sammons Matthew,Wade Robert A.

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference13 articles.

1. Discovery of (3S,3aR)-2-(3-Chloro-4-cyanophenyl)-3-cyclopentyl-3,3a,4,5-tetrahydro-2H-benzo[g]indazole-7-carboxylic Acid (PF-3882845), an Orally Efficacious Mineralocorticoid Receptor (MR) Antagonist for Hypertension and Nephropathy

2. An efficient synthesis and mechanism of formation of 6-acetyl-1,2-dihydro-2-oxo-3-pyridinecarboxylic acid

3. An efficient synthesis of 6-formyl-1,2-dihydro-2-oxo-3-pyridinecarboxylic acid and some carbonyl derivatives of it and its 6-acetyl homologue

4. Microwave-assisted cross-coupling of 3-chloro-2-pyrazolines and 3-chloro-1-phenyl-1,4,5,6-tetrahydropyridazine with aryl boronic acids

5. A Divergent Approach to the Synthesis of 3-Substituted-2-pyrazolines: Suzuki Cross-Coupling of 3-Sulfonyloxy-2-pyrazolines

Cited by 9 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. The 2‐Pyridyl Problem: Challenging Nucleophiles in Cross‐Coupling Arylations;Angewandte Chemie International Edition;2020-11-17

2. The 2‐Pyridyl Problem: Challenging Nucleophiles in Cross‐Coupling Arylations;Angewandte Chemie;2020-11-17

3. Isoxazole Strategy for the Synthesis of 2,2′-Bipyridine Ligands: Symmetrical and Unsymmetrical 6,6′-Binicotinates, 2,2′-Bipyridine-5-carboxylates, and Their Metal Complexes;The Journal of Organic Chemistry;2019-02-27

4. Csp2–Br bond activation of Br-pyridine by neophylpalladacycle: formation of binuclear seven-membered palladacycle and bipyridine species;New Journal of Chemistry;2017

5. Identification of (R)-6-(1-(4-Cyano-3-methylphenyl)-5-cyclopentyl-4,5-dihydro-1H-pyrazol-3-yl)-2-methoxynicotinic Acid, a Highly Potent and Selective Nonsteroidal Mineralocorticoid Receptor Antagonist;Journal of Medicinal Chemistry;2014-04-30