Pharmacological characterization of 17-cyclopropylmethyl-3,14-dihydroxy-4,5-epoxy-6-[(3′-fluoro-4′-pyridyl)acetamido]morphinan (NFP) as a dual selective MOR/KOR ligand with potential applications in treating opioid use disorder-Reference-Cited by-同舟云学术

Pharmacological characterization of 17-cyclopropylmethyl-3,14-dihydroxy-4,5-epoxy-6-[(3′-fluoro-4′-pyridyl)acetamido]morphinan (NFP) as a dual selective MOR/KOR ligand with potential applications in treating opioid use disorder

Published:2019-12 Issue: Volume:865 Page:172812
ISSN:0014-2999
Container-title:European Journal of Pharmacology
language:en
Short-container-title:European Journal of Pharmacology

Author:

Zheng Yi,Obeng Samuel,Reinecke Bethany A.,Chen Chongguang,Phansalkar Palak S.,Walentiny David M.,Gerk Phillip M.,Liu-Chen Lee-Yuan,Selley Dana E.,Beardsley Patrick M.,Zhang Yan

Funder

NIH/NIDA

Publisher

Elsevier BV

Subject

Pharmacology

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2. Verifying the role of 3-hydroxy of 17-cyclopropylmethyl-4,5α-epoxy-3,14β-dihydroxy-6β-[(4′-pyridyl) carboxamido]morphinan derivatives via their binding affinity and selectivity profiles on opioid receptors;Bioorganic Chemistry;2021-04

3. Stereoselective syntheses of 3-dehydroxynaltrexamines and N-methyl-3-dehydroxynaltrexamines;Tetrahedron Letters;2020-09