Validation of a conscious rat model for the discovery of novel agents that inhibit gastric acid secretion
Author:
Publisher
Elsevier BV
Subject
Pharmacology
Reference8 articles.
1. Application of a combined effect compartment and binding model for gastric acid inhibition of AR-HO47108: a potassium competitive acid blocker, and its active metabolite AR-HO47116 in the dog;Abelo;Eur. J. Pharm. Sci.,2006
2. A novel method of measurement of gastric acid secretion in intact and conscious rats;Hagiwara;Yakugaku. Zasshi.,1984
3. Animal pharmacology of reversible antagonism of the gastric acid pump, compared to standard antisecretory principles;Kromer;Pharmacology,2000
4. Properties of the reversible, K(+)-competitive inhibitor of the gastric (H+/K+)-ATPase, SK&F 97574. II. Pharmacological properties;Parsons;Biochem. Pharmacol.,1995
5. An explanation of gastric hypersecretion in the pylorus-ligated rat;Pober;Arch. Physiol. Biochem.,1999
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