Peripheral antinociceptive efficacy and potency of a novel opioid compound 14- O -MeM6SU in comparison to known peptide and non-peptide opioid agonists in a rat model of inflammatory pain-Reference-Cited by-同舟云学术

Peripheral antinociceptive efficacy and potency of a novel opioid compound 14- O -MeM6SU in comparison to known peptide and non-peptide opioid agonists in a rat model of inflammatory pain

Published:2013-08 Issue:1-3 Volume:713 Page:54-57
ISSN:0014-2999
Container-title:European Journal of Pharmacology
language:en
Short-container-title:European Journal of Pharmacology

Author:

Khalefa Baled. I.,Mousa Shaaban A.,Shaqura Mohammed,Lackó Erzsébet,Hosztafi Sándor,Riba Pál,Schäfer Michael,Ferdinandy Péter,Fürst Susanna,Al-Khrasani Mahmoud

Publisher

Elsevier BV

Subject

Pharmacology

Reference23 articles.

1. Receptor constants for endomorphin-1 and endomprphin-1-ol indicate differences in efficacy and receptor occupancy;Al Khrasani;Eur. J. Pharmacol.,2001

2. DAMGO and 6 beta-glycine substituted 14-O-methyloxymorphone but not morphine show peripheral, preemptive antinociception after systemic administration in a mouse visceral pain model and high intrinsic efficacy in the isolated rat vas deferens;Al Khrasani;Brain Res. Bull.,2007

3. Perineurial defect and peripheral opioid analgesia in inflammation;Antonijevic;J. Neurosci.,1995

4. Endogenous peripheral antinociception in early inflammation is not limited by the number of opioid-containing leukocytes but by opioid receptor expression;Brack;Pain,2004

5. Beta-endorphin—analgesic and hormonal effects in humans;Foley;Proc. Natl. Acad. Sci. U.S.A.,1979

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