Novel analgesic agents obtained by molecular hybridization of orthosteric and allosteric ligands
Author:
Publisher
Elsevier BV
Subject
Pharmacology
Reference36 articles.
1. Dualsteric GPCR targeting: a novel route to binding and signaling pathway selectivity;Antony;Faseb. J.,2009
2. New analogues of oxotremorine and oxotremorine-M: estimation of their in vitro affinity and efficacy at muscarinic receptor subtypes;Barocelli;Life Sci.,2000
3. Evidence for specific analgesic activity of a muscarinic agonist selected among a new series of acetylenic derivatives;Barocelli;Life Sci.,2001
4. Ligand binding enS.E.M.bles determine graded agonist efficacies at a G protein-coupled receptor;Bock;J. Biol. Chem.,2016
5. The allosteric vestibule of a seven transmembrane helical receptor controls G-protein coupling;Bock;Nat. Commun.,2012
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