N-Butyl-N-methyl-11-(3'-hydroxy-21',17'-carbolactone-19'-nor-17'α-pregna-1',3',5'(10')-trien-7'α-yl)-undecanamide: an inhibitor of type 2 17β-hydroxysteroid dehydrogenase that does not have oestrogenic or androgenic activity-Reference-Cited by-同舟云学术

N-Butyl-N-methyl-11-(3'-hydroxy-21',17'-carbolactone-19'-nor-17'α-pregna-1',3',5'(10')-trien-7'α-yl)-undecanamide: an inhibitor of type 2 17β-hydroxysteroid dehydrogenase that does not have oestrogenic or androgenic activity

Published:2000-02 Issue:2 Volume:35 Page:217-225
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Sam Kay-Mane,Labrie Fernand,Poirier Donald

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference44 articles.

1. The key role of 17β-hydroxysteroid dehydrogenases in sex steroid biology

2. 17β-Hydroxysteroid Dehydrogenases: Physiological Roles in Health and Disease

3. 17 -Hydroxysteroid dehydrogenase: inhibitors and inhibitor design

4. Intracrinology

5. A 6β-(thiaheptanamide) derivative of estradiol as inhibitor of 17β-hydroxysteroid dehydrogenase type 1

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