Development and application of a physiologically based pharmacokinetic model for entrectinib in rats and scale-up to humans: Route-dependent gut wall metabolism-Reference-Cited by-同舟云学术

Development and application of a physiologically based pharmacokinetic model for entrectinib in rats and scale-up to humans: Route-dependent gut wall metabolism

Published:2022-02 Issue: Volume:146 Page:112520
ISSN:0753-3322
Container-title:Biomedicine & Pharmacotherapy
language:en
Short-container-title:Biomedicine & Pharmacotherapy

Author:

Seo Seong-Wook,Han Dong-Gyun,Choi Eugene,Park Taeuk,Byun Jong Hyuk,Cho Hyun-Jong,Jung Il Hyo,Yoon In-Soo

Funder

National Research Foundation of Korea

Ministry of Science and ICT, South Korea

Publisher

Elsevier BV

Subject

Pharmacology,General Medicine

Reference51 articles.

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4. Activity of entrectinib in a patient with the first reported NTRK fusion in neuroendocrine cancer;Sigal;J. Natl. Compr. Canc. Netw.,2017

5. Physiologically based absorption modelling to explore the impact of food and gastric pH changes on the pharmacokinetics of entrectinib;Parrott;AAPS J.,2020

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