Slow binding–tight binding interaction between benzimidazol-2-one inhibitors and HIV-1 reverse transcriptase containing the lysine 103 to asparagine mutation
Author:
Publisher
Elsevier BV
Subject
Virology,Pharmacology
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1. I2-Mediated transition-metal-free aromatic C–H amination for the synthesis of benzimidazol-2-ones and related heterocycles;New Journal of Chemistry;2018
2. 2D and 3D QSAR of Benzimidazole Analogues as Novel HIV-1 Non Nucleoside Reverse Transcriptase Inhibitors;Indian Journal of Pharmaceutical Education and Research;2017-05-01
3. Drug Discoveries and Molecular Mechanism of Action;Successful Drug Discovery;2015-01-30
4. Design and synthesis of N1-aryl-benzimidazoles 2-substituted as novel HIV-1 non-nucleoside reverse transcriptase inhibitors;Bioorganic & Medicinal Chemistry;2014-02
5. Synthesis, Biological Activity, and ADME Properties of Novel S-DABOs/N-DABOs as HIV Reverse Transcriptase Inhibitors;ChemMedChem;2012-03-14
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