Development of a potent and selective chemical probe for the pleiotropic kinase CK2-Reference-Cited by-同舟云学术

Development of a potent and selective chemical probe for the pleiotropic kinase CK2

Published:2021-04 Issue:4 Volume:28 Page:546-558.e10
ISSN:2451-9456
Container-title:Cell Chemical Biology
language:en
Short-container-title:Cell Chemical Biology

Author:

Wells Carrow I.,Drewry David H.^ORCID,Pickett Julie E.,Tjaden Amelie^ORCID,Krämer Andreas,Müller Susanne,Gyenis Laszlo^ORCID,Menyhart Daniel^ORCID,Litchfield David W.,Knapp Stefan,Axtman Alison D.^ORCID

Funder

U.S. Department of Defense

Natural Sciences and Engineering Research Council of Canada

North Carolina Biotechnology Center

National Institutes of Health

Canadian Institutes of Health Research

Publisher

Elsevier BV

Subject

Clinical Biochemistry,Drug Discovery,Pharmacology,Molecular Biology,Molecular Medicine,Biochemistry

Reference72 articles.

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4. Inhibition of dual-specificity tyrosine phosphorylation-regulated kinase 2 perturbs 26S proteasome-addicted neoplastic progression;Banerjee;Proc. Natl. Acad. Sci. U S A,2019

5. Unprecedented selectivity and structural determinants of a new class of protein kinase CK2 inhibitors in clinical trials for the treatment of cancer;Battistutta;Biochemistry,2011

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