Synthesis of {1-[2′,5′-Bis-O-(t-butyldimethylsilyl)-β-d-xylo- and β-d-ribofuranosyl]thymine}-3′-spiro-5″-{4″-amino-1″,2″-oxathiole-2″,2″-dioxide} (TSAO). A novel type of specific anti-HIV agents-Reference-Cited by-同舟云学术

Synthesis of {1-[2′,5′-Bis-O-(t-butyldimethylsilyl)-β-d-xylo- and β-d-ribofuranosyl]thymine}-3′-spiro-5″-{4″-amino-1″,2″-oxathiole-2″,2″-dioxide} (TSAO). A novel type of specific anti-HIV agents

Published:1992-05 Issue:21 Volume:33 Page:3029-3032
ISSN:0040-4039
Container-title:Tetrahedron Letters
language:en
Short-container-title:Tetrahedron Letters

Author:

Pérez-Pérez María-Jesús,San-Félix Ana,María-José Camarasa,Balzarini Jan,Erik de Clercq

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference18 articles.

1. AZT Collaborative Working Group;Fischl;New Engl. J. Med.,1987

2. Anti-retroviral therapy of AIDS and related disorders: General principles and specific development of dideoxynucleosides

3. In Vivo Activity Against HIV and Favorable Toxicity Profile of 2′,3′-Dideoxyinosine

4. The Toxicity of Azidothymidine (AZT) in the Treatment of Patients with AIDS and AIDS-Related Complex

Cited by 44 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. A brief survey on the application of metal-catalyzed azide–alkyne cycloaddition reactions to the synthesis of ferrocenyl-x-1,2,3-triazolyl-R (x = none or a linker and R = organic entity) compounds with anticancer activity;Coordination Chemistry Reviews;2023-03

2. Cyanohydrins and Aminocyanides as Key Intermediates to Various Spiroheterocyclic Sugars;Topics in Heterocyclic Chemistry;2019

3. Preparation of Spiro[4.4]oxaphospholene and -azaphospholene Systems from Carbohydrate Templates;The Journal of Organic Chemistry;2013-08-29

4. Synthesis and in vitro activity of novel N-3 acylated TSAO-T compounds against HIV-1 and HCV;European Journal of Medicinal Chemistry;2011-10

5. Synthesis and characterization of new 1,4 and 1,5-disubstituted glucopyranosyl 1,2,3-triazole by 1,3-dipolar cycloaddition;Journal of Molecular Structure;2009-07