Dipeptide isosteres. 2. Synthesis of hydroxyethylene dipeptide isostere diastereomers from a common γ-lactone intermediate. Preparation of renin and HIV-1 protease inhibitor transition state mimics.-Reference-Cited by-同舟云学术

Dipeptide isosteres. 2. Synthesis of hydroxyethylene dipeptide isostere diastereomers from a common γ-lactone intermediate. Preparation of renin and HIV-1 protease inhibitor transition state mimics.

Published:1993-01 Issue:39 Volume:49 Page:8739-8756
ISSN:0040-4020
Container-title:Tetrahedron
language:en
Short-container-title:Tetrahedron

Author:

Baker William R.,Pratt John K.

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference45 articles.

1. C-Terminal modifications of nonpeptide renin inhibitors: improved oral bioavailability via modification of physicochemical properties

2. Benzocycloalkyl amines as novel C-termini for HIV protease inhibitors

3. Synthetic and enzyme inhibition studies of pepstatin analogs containing hydroxyethylene and ketomethylene dipeptide isosteres

4. Stereocontrolled addition of chiral, non-racemic amide homoenolates to t-Boc-(S)-phenylalaninal

Cited by 48 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. My 50-Plus Years of Academic Research Collaborations with Industry. A Retrospective;The Journal of Organic Chemistry;2024-06-12

2. Repurposed Antiviral Drugs for the Treatment of COVID-19: Syntheses, Mechanism of Infection and Clinical Trials;Mini-Reviews in Medicinal Chemistry;2021-05-19

3. Cross-Coupling of Ketone Enolates with Grignard and Zinc Reagents with First-Row Transition Metal Catalysts;ACS Catalysis;2021-04-27

4. Synthesis of anti-1,3 Amino Alcohol Motifs via Pd(II)/SOX Catalysis with the Capacity for Stereodivergence;Journal of the American Chemical Society;2019-05-29

5. Base-Mediated Tandem Reaction of α-Aryloxyacetophenones with Phosphonates: Selective Synthesis of Enol Phosphates;Synthesis;2012-02-17