Subergorgic acid, a novel tricyclopentanoid cardiotoxin from the pacific gorgonian coral

Author:

Groweiss Amiram,Fenical William,Cun-heng He,Clardy Jon,Zhongde Wu,Zhongnian Yiao,Kanghou Long

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference10 articles.

1. In addition, the pregnane steroids Δ1-pregnene-3βol-20-one, Δ4-pregnene-3,20-dione, Δ4-pregnene-3βol-20-one, and Δ1,4-pregnadiene-3,20-dione were isolated.

2. For subergorgic acid (1): m.p. 179–180°; [α]D -230° (c. 0.7, CHCl3); 1H NMR (360 MHz, CDCl3): δ 6.43 (1H, bs, C-9), 3.01 (1H, q, J=7 Hz, C-11), 2.37 (1H, dd, J=16.7, 6.7, C-3), 2.09 (1H, dd, J=8.8, 6.7, C-5), 2.01 (1H, dd, J=16.7, 12.6. C-3), 1.22 (3H, s, C-13), 1.13 (3H, d, J=7.3, C-15), 1.12 (3Hd, J=6.4C-12); 13C NMR (50 MHz, CDCl3): δ217.8 (s, C-2), 169.6 (s, C-14), 152.1 (d, C-9), 136.6 (s, C-10), 68.5 (s, C-1), 61.7 (s, C-8), 62.6, 51.6, 33.3 (all d's, C-4, C-5, and C-11), 49.9, 38.2, 28.3 (all t's, C-3, C-6, and C-7), 23.4, 19.9, 17.7 (all q's, C-12, C-13, and C-15); HRMS (EI): M+ m/z=248.1405 (26%), M+-H2O 230.1332 (100%), 215.1118 (29%), M+-COOH 203.1443 (27%), 202 (30%); IR (CH2Cl2): 1730. 1690, and 1645 cm-1.

3. For methyl ester 2: 1H NMR (CDCl3): δ 6.28 (1H, s, C-9), 3.73 (3H, s, OMe), 3.02 (1H, q, J=7.1, C-11), 2.35 (1H, dd, J=16.6, 6.8, C-3), 2.08 (1H, dd, J=8.9, 6.8, C-5), 2.00 (1H, dd, J=16.6, 12.6, C-3), 1.20 (3H, s, C-13), 1.12 (3H, d, J=6.4, C-12), 1.11 (3H, d, J=7.1, C-15); IR (CCl4): 1730, 1710, 1650, 1540, 1520, 1490, and 1460 cm−1.

4. For alcohol 3: 1H NMR (360 MHz, CDCl3): δ 5.14 (1H, s, C-9), 4.18 (3H, m, C-2 and C-14), 2.76 (1H, q, J=7, C-11), 1.93 (1H, ddd, J=15, 10, 4, C-3), 1.30 (3H, d, J=7, C-15), 1.15 (3H, s, C-13), 1.13 (3H, d, J=6.6, C-12); IR (CCl4): 3600, 1640, 1540, 1520, 1500, and 1450 cm−1. For alcohol 4: 1H NMR (CDCl3): δ 5.25 (1H, s, C-9), 4.36 (1H, bs, C-2), 4.15 (2H, AB q, J=13.4, C-14), 2.36 (1H. q, J=7, C-11), 1.33 (3H, s, C-13). 1.05 (3H, d, J=7, C-15), 1.04 (3H, d, J=6.4, C-12); IR (CCl4): 3600, 1640, 1540, 1510, 1490, and 1450 cm−1. The stereochemistries of 3 and 4 were based on the downfield shift of the 1H NMR signal of C-13 in 4 and the similar shift of C-15 in 3.

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号  京ICP备18003416号-3