Initial Structure–Activity Relationship Studies of a Novel Series of Pyrrolo[1,2-a]pyrimid-7-ones as GnRH Receptor Antagonists-Reference-Cited by-同舟云学术

Initial Structure–Activity Relationship Studies of a Novel Series of Pyrrolo[1,2-a]pyrimid-7-ones as GnRH Receptor Antagonists

Published:2002-02 Issue:3 Volume:12 Page:399-402
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Zhu Yun-Fei,Struthers R.Scott,Connors, Jr. Patrick J.,Gao Yinghong,Gross Timothy D.,Saunders John,Wilcoxen Keith,Reinhart Greg J.,Ling Nicholas,Chen Chen

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference15 articles.

1. Structure of the porcine LH- and FSH-releasing hormone. I. The proposed amino acid sequence

2. Primary Structure of the Ovine Hypothalamic Luteinizing Hormone-Releasing Factor (LRF)

3. Synthetic analogs of luteinizing hormone releasing hormone (LH-RH) substituted in position 6 and 10

4. Discovery of a Novel, Potent, and Orally Active Nonpeptide Antagonist of the Human Luteinizing Hormone-Releasing Hormone (LHRH) Receptor

5. Identification and initial structure-activity relationships of a novel non-peptide quinolone GnRH receptor antagonist

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