Dermorphin sequence with high δ-afinity by fixing the phe sidechain to trans at ξ1-Reference-Cited by-同舟云学术

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Dermorphin sequence with high δ-afinity by fixing the phe sidechain to trans at ξ1

Published:1992-10 Issue:10 Volume:2 Page:1305-1308
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Tourwé D.,Verschueren K.,Van Binst G.,Davis P.,Porreca F.,Hruby V.J.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference18 articles.

1. Deltorphins: a family of naturally occurring peptides with high affinity and selectivity for delta opioid binding sites.

2. Conformation-Activity relationships of cyclic dermorphin analogues

3. Conformational features responsible for the binding of cyclic analogues of enkephalin to opioid receptors III. Probable binding conformations of μ-agonists with phenylalanine in position 3

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1. Design, Synthesis, and In Vitro Characterization of Proteolytically-Stable Opioid-Neurotensin Hybrid Peptidomimetics;ACS Pharmacology & Translational Science;2024-08-19

2. χ-Space Screening of Dermorphin-Based Tetrapeptides through Use of Constrained Arylazepinone and Quinolinone Scaffolds;ACS Medicinal Chemistry Letters;2017-10-09

3. Side Chain Cyclized Aromatic Amino Acids: Great Tools as Local Constraints in Peptide and Peptidomimetic Design;Journal of Medicinal Chemistry;2016-10-12

4. Bifunctional Peptide-Based Opioid Agonist–Nociceptin Antagonist Ligands for Dual Treatment of Acute and Neuropathic Pain;Journal of Medicinal Chemistry;2016-04-14

5. 7-endo cyclization of 2,3-epoxyamides and 2,3-aziridine carboxamides by intramolecular Friedel–Crafts reaction;Tetrahedron: Asymmetry;2015-02

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