Synthesis and structure–activity relationships of 4-oxo-1-phenyl-3,4,6,7-tetrahydro-[1,4]diazepino[6,7,1- hi ]indoles: novel PDE4 inhibitors-Reference-Cited by-同舟云学术

Synthesis and structure–activity relationships of 4-oxo-1-phenyl-3,4,6,7-tetrahydro-[1,4]diazepino[6,7,1- hi ]indoles: novel PDE4 inhibitors

Published:2000-01 Issue:1 Volume:10 Page:35-38
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Pascal Yves,Andrianjara Charles R,Auclair Eric,Avenel Nadine,Bertin Bernadette,Calvet Alain,Féru Frédéric,Lardon Sophie,Moodley Indres,Ouagued Malika,Payne Adrian,Pruniaux Marie-Pierre,Szilagyi Corinne

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference14 articles.

1. Cyclic nucleotide phosphodiesterases: functional implications of multiple isoforms

2. Phosphodiesterase type IV inhibitors as antiinflammatory agents

3. Selective Inhibitors of Cyclic AMP-Specific Phosphodiesterase: Heterocycle-Condensed Purines

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