Synthesis and activity studies of conformationally restricted α-ketoamide factor Xa inhibitors-Reference-Cited by-同舟云学术

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Synthesis and activity studies of conformationally restricted α-ketoamide factor Xa inhibitors

Published:2000-06 Issue:11 Volume:10 Page:1253-1256
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Cacciola Joseph,Fevig John M.,Stouten Pieter F.W.,Alexander Richard S.,Knabb Robert M.,Wexler Ruth R.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference11 articles.

1. Synthesis of conformationally-restricted boropeptide thrombin inhibitors

2. Assays were performed as described in: Kettner, C.; Mersinger, L.; Knabb, R. J. Biol. Chem. 1990, 265, 18289.

3. Amide and α-keto carbonyl inhibitors of thrombin based on arginine and lysine: Synthesis, stability and biological characterization

4. The synthesis of lysine α-ketoamide thrombin inhibitord via an epoxy amide ring opening

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2. Development of Trypsin-Like Serine Protease Inhibitors as Therapeutic Agents: Opportunities, Challenges, and their Unique Structure-Based Rationales;Current Topics in Medicinal Chemistry;2016-03-01

3. Synthesis of β-amino-α.-ketoamides;Current Organic Chemistry;2014-10-21

4. Direct synthesis of the arylboronic acid analogues of phenylglycine via microwave-assisted four-component Ugi reaction;Tetrahedron;2014-03

5. The syntheses of α-ketoamides vianBu4NI-catalyzed multiple sp3C–H bond oxidation of ethylarenes and sequential coupling with dialkylformamides;Org. Biomol. Chem.;2014

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