Ether modifications to 1-[2-(3,4-dimethoxyphenyl)ethyl]-4-(3-phenylpropyl)piperazine (SA4503): Effects on binding affinity and selectivity for sigma receptors and monoamine transporters-Reference-Cited by-同舟云学术

Ether modifications to 1-[2-(3,4-dimethoxyphenyl)ethyl]-4-(3-phenylpropyl)piperazine (SA4503): Effects on binding affinity and selectivity for sigma receptors and monoamine transporters

Published:2015-01 Issue:1 Volume:23 Page:222-230
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Xu Rong,Lord Sarah A.,Peterson Ryan M.,Fergason-Cantrell Emily A.,Lever John R.,Lever Susan Z.

Funder

National Cancer Institute

National Institute for Drug Abuse

National Science Foundation

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference66 articles.

1. Sigma Receptors in Oncology: Therapeutic and Diagnostic Applications of Sigma Ligands

2. Sigma receptors and their ligands in cancer biology: overview and new perspectives for cancer therapy

3. The σ2 Receptor: A Novel Protein for the Imaging and Treatment of Cancer

4. Targeting ligand-operated chaperone sigma-1 receptors in the treatment of neuropsychiatric disorders

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