2-Aryladenine derivatives as a potent scaffold for A1, A3 and dual A1/A3 adenosine receptor antagonists: Synthesis and structure-activity relationships-Reference-Cited by-同舟云学术

2-Aryladenine derivatives as a potent scaffold for A1, A3 and dual A1/A3 adenosine receptor antagonists: Synthesis and structure-activity relationships

Published:2019-08 Issue:16 Volume:27 Page:3551-3558
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Areias Filipe,Correia Carla,Rocha Ashly,Brea José,Castro Marián,Loza Maria I.,Proença M. Fernanda,Carvalho M. Alice

Funder

Ministry of Science and Innovation

Xunta de Galicia

Carlos III Health Institute

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference19 articles.

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3. International Union of Basic and Clinical Pharmacology. LXXXI. Nomenclature and Classification of Adenosine Receptors—An Update

4. Introduction to adenosine receptors as therapeutic targets;Jacobson;Hand Exp Pharmacol,2009

5. Recent developments in adenosine receptor ligands and their potential as novel drugs;Muller;BBA,1808

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1. 2-Aryladenine Derivatives as a Potent Scaffold for Adenosine Receptor Antagonists: The 6-Morpholino Derivatives;Molecules;2024-05-28

2. Design, Synthesis and Biological Evaluation of 1,3,5-Triazine Derivatives Targeting hA1 and hA3 Adenosine Receptor;Molecules;2022-06-22

3. Pharmacological characterisation of novel adenosine A3 receptor antagonists;Scientific Reports;2020-11-27

4. Synthesis of 2-(aminophenyl)adenine derivatives: a simple protocol using the classical iron powder/acetic acid reduction methodology;Canadian Journal of Chemistry;2020-03

5. Pharmacological Characterisation of Novel Adenosine Receptor A3R Antagonists;2019-07-10