Synthesis and in vivo evaluation of 18F-fluoroethyl GF120918 and XR9576 as positron emission tomography probes for assessing the function of drug efflux transporters-Reference-Cited by-同舟云学术

Synthesis and in vivo evaluation of 18F-fluoroethyl GF120918 and XR9576 as positron emission tomography probes for assessing the function of drug efflux transporters

Published:2011-01 Issue:2 Volume:19 Page:861-870
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Kawamura Kazunori,Yamasaki Tomoteru,Konno Fujiko,Yui Joji,Hatori Akiko,Yanamoto Kazuhiko,Wakizaka Hidekatsu,Ogawa Masanao,Yoshida Yuichiro,Nengaki Nobuki,Fukumura Toshimitsu,Zhang Ming-Rong

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference35 articles.

1. Role of transport proteins in drug absorption, distribution and excretion

2. Mammalian ABC Transporters in Health and Disease

3. Mammalian drug efflux transporters of the ATP binding cassette (ABC) family: an overview

4. Role of drug efflux transporters in the brain for drug disposition and treatment of brain diseases

5. Multidrug resistance in cancer: role of ATP–dependent transporters

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