Design, synthesis and biological activity of amidinobicyclic compounds (derivatives of DX-9065a) as factor Xa inhibitors: SAR study of S1 and aryl binding sites-Reference-Cited by-同舟云学术

Design, synthesis and biological activity of amidinobicyclic compounds (derivatives of DX-9065a) as factor Xa inhibitors: SAR study of S1 and aryl binding sites

Published:2004-05 Issue:9 Volume:12 Page:2099-2114
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Komoriya Satoshi,Kanaya Naoaki,Nagahara Takayasu,Yokoyama Asako,Inamura Kazue,Yokoyama Yukio,Katakura Shin-ichi,Hara Tsuyoshi

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference10 articles.

1. The ideal anti-thrombotic drug

2. Dibasic (Amidinoaryl)propanoic Acid Derivatives as Novel Blood Coagulation Factor Xa Inhibitors

3. X-ray Structure of Active Site-inhibited Clotting Factor Xa

4. Synthese antileukämischer Indolylvinyl-1-benzofurane und-benzo[b]thiophene

5. 348. The preparation of benziminazoles and benzoxazoles from Schiff's bases. Part II

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