Synthesis and biological evaluation of novel tyrosyl-DNA phosphodiesterase 1 inhibitors with a benzopentathiepine moiety-Reference-Cited by-同舟云学术

Synthesis and biological evaluation of novel tyrosyl-DNA phosphodiesterase 1 inhibitors with a benzopentathiepine moiety

Published:2015-05 Issue:9 Volume:23 Page:2044-2052
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Zakharenko Alexandra,Khomenko Tatyana,Zhukova Svetlana,Koval Olga,Zakharova Olga,Anarbaev Rashid,Lebedeva Natalya,Korchagina Dina,Komarova Nina,Vasiliev Vladimir,Reynisson Jóhannes,Volcho Konstantin,Salakhutdinov Nariman,Lavrik Olga

Funder

Ministry of Education and Science of Russian Federation

Russian Science Foundation

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference61 articles.

1. Base excision repair in the mammalian brain: Implication for age related neurodegeneration

2. The Therapeutic Potential of Poly(ADP-Ribose) Polymerase Inhibitors

3. DNA damage repair and cardiovascular diseases

4. A human 5′-tyrosyl DNA phosphodiesterase that repairs topoisomerase-mediated DNA damage

5. Tyrosyl-DNA phosphodiesterase I resolves both naturally and chemically induced DNA adducts and its potential as a therapeutic target

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