Fragment-based hit discovery and structure-based optimization of aminotriazoloquinazolines as novel Hsp90 inhibitors-Reference-Cited by-同舟云学术

Fragment-based hit discovery and structure-based optimization of aminotriazoloquinazolines as novel Hsp90 inhibitors

Published:2014-08 Issue:15 Volume:22 Page:4135-4150
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Casale Elena,Amboldi Nadia,Brasca Maria Gabriella,Caronni Dannica,Colombo Nicoletta,Dalvit Claudio,Felder Eduard R.,Fogliatto Gianpaolo,Galvani Arturo,Isacchi Antonella,Polucci Paolo,Riceputi Laura,Sola Francesco,Visco Carlo,Zuccotto Fabio,Casuscelli Francesco

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference55 articles.

1. Drugging the Cancer Chaperone HSP90: Combinatorial Therapeutic Exploitation of Oncogene Addiction and Tumor Stress

2. HSP90 and the chaperoning of cancer

3. Hsp90 Molecular Chaperone Inhibitors: Are We There Yet?

4. Preface to Hsp90

5. Advances in the clinical development of heat shock protein 90 (Hsp90) inhibitors in cancers

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