Design, synthesis and anti-tuberculosis activity of 1-adamantyl-3-heteroaryl ureas with improved in vitro pharmacokinetic properties-Reference-Cited by-同舟云学术

Design, synthesis and anti-tuberculosis activity of 1-adamantyl-3-heteroaryl ureas with improved in vitro pharmacokinetic properties

Published:2013-05 Issue:9 Volume:21 Page:2587-2599
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

North E. Jeffrey,Scherman Michael S.,Bruhn David F.,Scarborough Jerrod S.,Maddox Marcus M.,Jones Victoria,Grzegorzewicz Anna,Yang Lei,Hess Tamara,Morisseau Christophe,Jackson Mary,McNeil Michael R.,Lee Richard E.

Funder

National Institutes of Health

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference19 articles.

1. Global tuberculosis control: lessons learnt and future prospects

2. The structure–activity relationship of urea derivatives as anti-tuberculosis agents

3. EPOXIDE HYDROLASES: Mechanisms, Inhibitor Designs, and Biological Roles

4. The Molecular Structure of Epoxide Hydrolase B from Mycobacterium tuberculosis and Its Complex with a Urea-Based Inhibitor

5. Inhibition of mycolic acid transport across the Mycobacterium tuberculosis plasma membrane

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