Antagonists of the human A2A receptor. Part 6: Further optimization of pyrimidine-4-carboxamides-Reference-Cited by-同舟云学术

Antagonists of the human A2A receptor. Part 6: Further optimization of pyrimidine-4-carboxamides

Published:2009-09 Issue:18 Volume:17 Page:6590-6605
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Gillespie Roger J.,Bamford Samantha J.,Clay Alex,Gaur Suneel,Haymes Tim,Jackson Philip S.,Jordan Allan M.,Klenke Burkhard,Leonardi Stefania,Liu Jeanette,Mansell Howard L.,Ng Sean,Saadi Mona,Simmonite Heather,Stratton Gemma C.,Todd Richard S.,Williamson Douglas S.,Yule Ian A.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference23 articles.

1. Therapeutic potential of adenosine A2A receptor antagonists in Parkinson's disease

2. Adenosine A2Areceptor antagonist treatment of Parkinson’s disease

3. Antagonists of the human A2A receptor. Part 5: Highly bio-available pyrimidine-4-carboxamides

4. KW-6002

5. Adenosine A2Areceptor antagonist istradefylline (KW-6002) reduces “off” time in Parkinson's disease: A double-blind, randomized, multicenter clinical trial (6002-US-005)

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