A fragment-based approach leading to the discovery of a novel binding site and the selective CK2 inhibitor CAM4066-Reference-Cited by-同舟云学术

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A fragment-based approach leading to the discovery of a novel binding site and the selective CK2 inhibitor CAM4066

Published:2017-07 Issue:13 Volume:25 Page:3471-3482
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

De Fusco Claudia,Brear Paul,Iegre Jessica,Georgiou Kathy Hadje,Sore Hannah F.,Hyvönen Marko,Spring David R.

Funder

Wellcome Trust

European Research Council

Seventh Framework Programme

Engineering and Physical Sciences Research Council

Biotechnology and Biological Sciences Research Council

Medical Research Council

Royal Society

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference32 articles.

1. The rise of fragment-based drug discovery

2. Fragment-based lead discovery: leads by design

3. Fragment-based approaches to enzyme inhibition

4. Fragment-Based Approaches in Drug Discovery and Chemical Biology

5. Fragment Deconstruction of Small, Potent Factor Xa Inhibitors: Exploring the Superadditivity Energetics of Fragment Linking in Protein-Ligand Complexes

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1. Synthesis and evaluation of chemical linchpins for highly selective CK2α targeting;European Journal of Medicinal Chemistry;2024-10

2. Synthesis and evaluation of chemical linchpins for highly selective CK2α targeting;2024-05-16

3. Recent Advances in the Discovery of CK2 Inhibitors;ACS Omega;2024-05-03

4. CK2 Inhibitors Targeting Inside and Outside the Catalytic Box;Kinases and Phosphatases;2024-03-26

5. Anion cascade reactions III: Synthesis of 3-isoquinuclidone bridged polycyclic lactams;Chinese Chemical Letters;2024-02

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