Human HDAC isoform selectivity achieved via exploitation of the acetate release channel with structurally unique small molecule inhibitors-Reference-Cited by-同舟云学术

Human HDAC isoform selectivity achieved via exploitation of the acetate release channel with structurally unique small molecule inhibitors

Published:2011-08 Issue:15 Volume:19 Page:4626-4634
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Whitehead Lewis,Dobler Markus R.,Radetich Branko,Zhu Yanyi,Atadja Peter W.,Claiborne Tavina,Grob Jonathan E.,McRiner Andrew,Pancost Margaret R.,Patnaik Anup,Shao Wenlin,Shultz Michael,Tichkule Ritesh,Tommasi Ruben A.,Vash Brian,Wang Ping,Stams Travis

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference51 articles.

1. Conformational Refinement of Hydroxamate-Based Histone Deacetylase Inhibitors and Exploration of 3-Piperidin-3-ylindole Analogues of Dacinostat (LAQ824)

2. Deacetylase Enzymes

3. Histone deacetylases and cancer: causes and therapies

4. Human HDAC1 and HDAC2 function in the DNA-damage response to promote DNA nonhomologous end-joining

5. Histone Deacetylase: A Target for Antiproliferative and Antiprotozoal Agents

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