N-4-t-Butylbenzyl 2-(4-methylsulfonylaminophenyl) propanamide TRPV1 antagonists: Structure–activity relationships in the A-region-Reference-Cited by-同舟云学术

N-4-t-Butylbenzyl 2-(4-methylsulfonylaminophenyl) propanamide TRPV1 antagonists: Structure–activity relationships in the A-region

Published:2012-01 Issue:1 Volume:20 Page:215-224
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Kim Yong Soo,Kil Min-Jung,Kang Sang-Uk,Ryu HyungChul,Kim Myeong Seop,Cho Yongsung,Bhondwe Rahul S.,Thorat Shivaji A.,Sun Wei,Liu Keliang,Lee Jin Hee,Choi Sun,Pearce Larry V.,Pavlyukovets Vladimir A.,Morgan Matthew A.,Tran Richard,Lazar Jozsef,Blumberg Peter M.,Lee Jeewoo

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference20 articles.

1. The Cloned Capsaicin Receptor Integrates Multiple Pain-Producing Stimuli

2. The capsaicin receptor: a heat-activated ion channel in the pain pathway

3. Vanilloid receptors on sensory nerves mediate the vasodilator action of anandamide

4. Direct activation of capsaicin receptors by products of lipoxygenases: Endogenous capsaicin-like substances

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