α-Methylated simplified resiniferatoxin (sRTX) thiourea analogues as potent and stereospecific TRPV1 antagonists-Reference-Cited by-同舟云学术

α-Methylated simplified resiniferatoxin (sRTX) thiourea analogues as potent and stereospecific TRPV1 antagonists

Published:2014-06 Issue:12 Volume:24 Page:2685-2688
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Kim Ho Shin,Jin Mi-Kyoung,Kang Sang-Uk,Lim Ju-Ok,Tran Phuong-Thao,Hoang Van-Hai,Ann Jihyae,Ha Tae-Hwan,Pearce Larry V.,Pavlyukovets Vladimir A.,Blumberg Peter M.,Lee Jeewoo

Funder

National Research Foundation of Korea

Intramural Research Program of NIH

Center for Cancer Research

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference19 articles.

1. Capsazepine: a competitive antagonist of the sensory neurone excitant capsaicin

2. High Affinity Antagonists of the Vanilloid Receptor

3. Analgesic potential of TRPV1 antagonists

4. Therapeutic potential of vanilloid receptor TRPV1 agonists and antagonists as analgesics: Recent advances and setbacks

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