Discovery of novel, highly potent and selective β-hairpin mimetic CXCR4 inhibitors with excellent anti-HIV activity and pharmacokinetic profiles-Reference-Cited by-同舟云学术

Discovery of novel, highly potent and selective β-hairpin mimetic CXCR4 inhibitors with excellent anti-HIV activity and pharmacokinetic profiles

Published:2006-12 Issue:24 Volume:14 Page:8396-8404
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

DeMarco Steven J.,Henze Heiko,Lederer Alexander,Moehle Kerstin,Mukherjee Reshmi,Romagnoli Barbara,Robinson John A.,Brianza Federico,Gombert Frank O.,Lociuro Sergio,Ludin Christian,Vrijbloed Jan Willem,Zumbrunn Jürg,Obrecht Jean-Pierre,Obrecht Daniel,Brondani Vincent,Hamy François,Klimkait Thomas

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference49 articles.

1. Substitutions in a Homologous Region of Extracellular Loop 2 of CXCR4 and CCR5 Alter Coreceptor Activities for HIV-1 Membrane Fusion and Virus Entry

2. HIV-1 Entry Cofactor: Functional cDNA Cloning of a Seven-Transmembrane, G Protein-Coupled Receptor

3. New targets for inhibitors of HIV-1 replication

4. CC CKR5: A RANTES, MIP-1α, MIP-1β Receptor as a Fusion Cofactor for Macrophage-Tropic HIV-1

5. HIV-1 entry into CD4+ cells is mediated by the chemokine receptor CC-CKR-5

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