Discovery and optimization of pyrrolo[1,2-a]pyrazinones leads to novel and selective inhibitors of PIM kinases-Reference-Cited by-同舟云学术

Discovery and optimization of pyrrolo[1,2-a]pyrazinones leads to novel and selective inhibitors of PIM kinases

Published:2013-12 Issue:23 Volume:21 Page:7364-7380
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Casuscelli Francesco,Ardini Elena,Avanzi Nilla,Casale Elena,Cervi Giovanni,D’Anello Matteo,Donati Daniele,Faiardi Daniela,Ferguson Ronald D.,Fogliatto Gianpaolo,Galvani Arturo,Marsiglio Aurelio,Mirizzi Danilo G.,Montemartini Marisa,Orrenius Christian,Papeo Gianluca,Piutti Claudia,Salom Barbara,Felder Eduard R.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference68 articles.

1. Mice Deficient for All PIM Kinases Display Reduced Body Size and Impaired Responses to Hematopoietic Growth Factors

2. For better or for worse: the role of Pim oncogenes in tumorigenesis

3. PIM serine/threonine kinases in the pathogenesis and therapy of hematologic malignancies and solid cancers

4. Pim kinases in cancer: Diagnostic, prognostic and treatment opportunities

5. Abnormal hematopoietic phenotypes in Pim kinase triple knockout mice

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