Synthesis and biological activity of selenopsammaplin A and its analogues as antitumor agents with DOT1L inhibitory activity-Reference-Cited by-同舟云学术

Synthesis and biological activity of selenopsammaplin A and its analogues as antitumor agents with DOT1L inhibitory activity

Published:2021-04 Issue: Volume:35 Page:116072
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Ju Han Hae,Sub Byun Woong,Ho Lee Gyu,Kyung Kim Won,Jang Kyungkuk,Yang Sehun,Yang Jewon,Woo Ha Min,Hong Suckchang,Lee Jeeyeon,Shin Jongheon,Bong Oh Ki,Kook Lee Sang,Park Hyeung-geun

Funder

National Research Foundation of Korea

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference44 articles.

1. The diverse functions of Dot1 and H3K79 methylation

2. Selective Inhibitors of Histone Methyltransferase DOT1L: Design, Synthesis, and Crystallographic Studies

3. MLL-Rearranged Leukemia Is Dependent on Aberrant H3K79 Methylation by DOT1L

4. DOT1L, the H3K79 methyltransferase, is required for MLL-AF9–mediated leukemogenesis

5. Selective Killing of Mixed Lineage Leukemia Cells by a Potent Small-Molecule DOT1L Inhibitor

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