In vitro and pharmacophore insights into CYP3A enzymes-Reference-Cited by-同舟云学术

In vitro and pharmacophore insights into CYP3A enzymes

Published:2003-04 Issue:4 Volume:24 Page:161-166
ISSN:0165-6147
Container-title:Trends in Pharmacological Sciences
language:en
Short-container-title:Trends in Pharmacological Sciences

Author:

Ekins Sean,Stresser David M.,Andrew Williams J.

Publisher

Elsevier BV

Subject

Pharmacology,Toxicology

Reference45 articles.

1. The human CYP3A subfamily: practical considerations;Wrighton;Drug Metab. Rev.,2000

2. Sequence diversity in CYP3A promotors and characterization of the genetic basis of polymorphic CYP3A5 expression;Kuehl;Nat. Genet.,2001

3. cDNA cloning and initial characterization of CYP3A43, a novel human cytochrome P450;Domanski;Mol. Pharmacol.,2001

4. Design and application of fluorimetric assays for human cytochrome P450 inhibition;Crespi;Methods Enzymol.,2002

5. Substrate-dependent modeulation of CYP3A4 catalytic activity: analysis of 27 test compounds with four fluorimetric substrates;Stresser;Drug Metab. Dispos.,2000

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