Pharmacokinetic–pharmacodynamic modelling of tiagabine CNS effects upon chronic treatment in rats: lack of change in concentration–EEG effect relationship-Reference-Cited by-同舟云学术

Pharmacokinetic–pharmacodynamic modelling of tiagabine CNS effects upon chronic treatment in rats: lack of change in concentration–EEG effect relationship

Published:2000-12 Issue:2 Volume:12 Page:141-150
ISSN:0928-0987
Container-title:European Journal of Pharmaceutical Sciences
language:en
Short-container-title:European Journal of Pharmaceutical Sciences

Author:

Cleton A.,Altorf B.A.,Voskuyl R.A.,Danhof M.

Publisher

Elsevier BV

Subject

Pharmaceutical Science

Reference30 articles.

1. Imidazenil, a partial positive allosteric modulator of GABAA receptors, exhibits low tolerance and dependence liabilities in the rat;Auta;J. Pharmacol. Exp. Ther.,1994

2. (R)-N-[4,4-Bis(3-methyl-2-thienyl)but-3-en-1-yl]nipecotic acid binds with high affinity to the brain γ-aminobutyric acid uptake carrier;Braestrup;J. Neurochem.,1990

3. Stereoselective central nervous system effects of the R- and S-isomers of the GABA uptake blocker N-(4,4-di-(3-methylthien-2-yl)but-3-enyl) nipecotic acid in the rat;Cleton;Br. J. Pharmacol.,1999

4. Mechanism-based modelling of adaptive changes in the pharmacodynamics of midazolam in the kindling model of epilepsy;Cleton;Pharm. Res.,1999

5. Effect of amygdala kindling on the central nervous system effects of tiagabine: EEG effects versus GABA levels;Cleton;Br. J. Pharmacol.,2000

Cited by 6 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Introduction: Utility of Mathematical Models in Drug Development and Delivery;Drug Delivery Approaches;2021-07-27

2. Facile One-Pot Synthesis of 1,2,3,4-Tetrahydroquinoline-3-carboxylic Acids and Their Heterocyclic Analogs;Synthetic Communications;2008-08-18

3. Effect of the administration of tiagabine and gabapentin on rabbit electroencephalogram activity;Journal of Pharmacy and Pharmacology;2006-10

4. From Neuroscience to Application in Neuropharmacology: A Generation of Progress in Electrophysiology;Clinical EEG and Neuroscience;2006-04

5. The interaction between vigabatrin and diazepam on the electroencephalogram during active behaviour in rats: an isobolic analysis;European Journal of Pharmacology;2004-07