Identification of harmine and β-carboline analogs from a high-throughput screen of an approved drug collection; profiling as differential inhibitors of DYRK1A and monoamine oxidase A and for in vitro and in vivo anti-cancer studies-Reference-Cited by-同舟云学术

Identification of harmine and β-carboline analogs from a high-throughput screen of an approved drug collection; profiling as differential inhibitors of DYRK1A and monoamine oxidase A and for in vitro and in vivo anti-cancer studies

Published:2021-07 Issue: Volume:162 Page:105821
ISSN:0928-0987
Container-title:European Journal of Pharmaceutical Sciences
language:en
Short-container-title:European Journal of Pharmaceutical Sciences

Author:

Tarpley Michael,Oladapo Helen O.,Strepay Dillon^ORCID,Caligan Thomas B.,Chdid Lhoucine,Shehata Hassan^ORCID,Roques Jose R.^ORCID,Thomas Rhashad,Laudeman Christopher P.^ORCID,Onyenwoke Rob U.,Darr David B.,Williams Kevin P.^ORCID

Funder

North Carolina Central University

Publisher

Elsevier BV

Subject

Pharmaceutical Science

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3. Harmine is an ATP-competitive inhibitor for dual-specificity tyrosine phosphorylation-regulated kinase 1A (Dyrk1A);Adayev;Arch Biochem Biophys,2011

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5. Beta-carbolines, psychoactive compounds in the mammalian body. Part I: Occurrence, origin and metabolism;Airaksinen;Med Biol,1981

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