Inhibition of ABCG2/BCRP-mediated transport–correlation analysis of various expression systems and probe substrates

Author:

Sáfár Zsolt,Kecskeméti GáborORCID,Molnár Judit,Kurunczi Anita,Szabó Zoltán,Janáky Tamás,Kis Emese,Krajcsi Péter

Publisher

Elsevier BV

Subject

Pharmaceutical Science

Reference35 articles.

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3. EMA, 2012. Guideline on the investigation of drug interactions. https://www.ema.europa.eu/documents/scientific-guideline/guideline-investigation-drug-interactions_en.pdf.

4. FDA, 2017. In Vitro Metabolism and Transporter Mediated Drug-Drug Interaction Studies Guidance for Industry. https://www.fda.gov/downloads/Drugs/GuidanceComplianceRegulatoryInformation/Guidances/UCM581965.pdf.

5. FDA, 2020. In vitro drug interaction studies — cytochrome P450 enzyme- and transporter-mediated drug interactions guidance for industry. https://www.fda.gov/media/134582/download.

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