Fragment Screening of Stabilized G-Protein-Coupled Receptors Using Biophysical Methods
Author:
Publisher
Elsevier
Reference22 articles.
1. An integrated approach to fragment-based lead generation: Philosophy, strategy and case studies from AstraZeneca's drug discovery programmes;Albert;Curr. Top. Med. Chem.,2007
2. Refolded outer membrane protein A of Escherichia coli forms ion channels with two conductance states in planar lipid bilayers;Arora;J. Biol. Chem.,2000
3. High-resolution crystal structure of an engineered human β2-adrenergic G protein-coupled receptor;Cherezov;Science,2007
4. From fragment to clinical candidate—A historical perspective;Chessari;Drug Discov. Today,2009
5. A ‘rule of three’ for fragment-based lead discovery?;Congreve;Drug Discov. Today,2003
Cited by 108 articles. 订阅此论文施引文献 订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献
1. Agonist Discovery for Membrane Proteins on Live Cells by Using DNA-encoded Libraries;Journal of the American Chemical Society;2024-08-22
2. Exploring the interactions of biologically active compounds (including drugs) with biomolecules: Utilizing Surface Plasmon Resonance and SwitchSense techniques;TrAC Trends in Analytical Chemistry;2024-07
3. Optimizing NMR fragment-based drug screening for membrane protein targets;Journal of Structural Biology: X;2024-06
4. Direct Binding Methods to Measure Receptor–Ligand Interactions;The Journal of Physical Chemistry B;2023-12-22
5. Extending the Affinity Range of Weak Affinity Chromatography for the Identification of Weak Ligands Targeting Membrane Proteins;Molecules;2023-10-16
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线，采集、加工和组织学术论文而形成的新型学术文献查询和分析系统，可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容，当前同舟云学术共收录了国内外主流学术期刊6万余种，收集的期刊论文及会议论文总量共计约1.5亿篇，并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询！咨询电话：010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3