Identification of potent and orally bioavailable nucleotide competing reverse transcriptase inhibitors: In vitro and in vivo optimization of a series of benzofurano[3,2-d]pyrimidin-2-one derived inhibitors-Reference-Cited by-同舟云学术

Identification of potent and orally bioavailable nucleotide competing reverse transcriptase inhibitors: In vitro and in vivo optimization of a series of benzofurano[3,2-d]pyrimidin-2-one derived inhibitors

Published:2013-07 Issue:13 Volume:23 Page:3967-3975
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Sturino Claudio F.,Bousquet Yves,James Clint A.,DeRoy Patrick,Duplessis Martin,Edwards Paul J.,Halmos Ted,Minville Joannie,Morency Louis,Morin Sébastien,Thavonekham Bounkham,Tremblay Martin,Duan Jianmin,Ribadeneira Maria,Garneau Michel,Pelletier Alex,Tremblay Sonia,Lamorte Louie,Bethell Richard,Cordingley Michael G.,Rajotte Daniel,Simoneau Bruno

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference34 articles.

1. The development of antiretroviral therapy and its impact on the HIV-1/AIDS pandemic

2. UNAIDS Report on the Global Aids Epidemic, 2012. See: http://www.unaids.org/en/media/unaids/contentassets/documents/epidemiology/2012/gr2012/20121120_UNAIDS_Global_Report_2012_en.pdf (Accessed: December 5, 2012).

3. HIV Co-receptors as Targets for Antiviral Therapy

4. Targeting CXCR4 in HIV Cell-Entry Inhibition.

5. The chemokine system and CCR5 antagonists: potential in HIV treatment and other novel therapies

Cited by 5 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. The anti-HIV potential of imidazole, oxazole and thiazole hybrids: A mini-review;Arabian Journal of Chemistry;2022-11

2. HIV nucleoside reverse transcriptase inhibitors;European Journal of Medicinal Chemistry;2022-10

3. Aligning Potency and Pharmacokinetic Properties for Pyridine-Based NCINIs;ACS Medicinal Chemistry Letters;2016-06-13

4. Subtype-Specific Analysis of the K65R Substitution in HIV-1 That Confers Hypersusceptibility to a Novel Nucleotide-Competing Reverse Transcriptase Inhibitor;Antimicrobial Agents and Chemotherapy;2015-03-16

5. Effects of the W153L Substitution in HIV Reverse Transcriptase on Viral Replication and Drug Resistance to Multiple Categories of Reverse Transcriptase Inhibitors;Antimicrobial Agents and Chemotherapy;2014-05-27