Identification of spirocyclic piperidine-azetidine inverse agonists of the ghrelin receptor-Reference-Cited by-同舟云学术

Identification of spirocyclic piperidine-azetidine inverse agonists of the ghrelin receptor

Published:2012-07 Issue:13 Volume:22 Page:4281-4287
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Kung Daniel W.,Coffey Steven B.,Jones Ryan M.,Cabral Shawn,Jiao Wenhua,Fichtner Michael,Carpino Philip A.,Rose Colin R.,Hank Richard F.,Lopaze Michael G.,Swartz Roger,(Tommy) Chen Hou,Hendsch Zachary,Posner Bruce,Wielis Christopher F.,Manning Brian,Dubins Jeffrey,Stock Ingrid A.,Varma Sam,Campbell Mary,DeBartola Demetria,Kosa-Maines Rachel,Steyn Stefanus J.,McClure Kim F.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference30 articles.

1. Ghrelin is a growth-hormone-releasing acylated peptide from stomach

2. Effects of an Oral Ghrelin Mimetic on Body Composition and Clinical Outcomes in Healthy Older Adults

3. Pyrazolinone-piperidine dipeptide growth hormone secretagogues (GHSs)

4. Optimization of the Potency and Pharmacokinetic Properties of a Macrocyclic Ghrelin Receptor Agonist (Part I): Development of Ulimorelin (TZP-101) from Hit to Clinic

5. Ghrelin and Energy Balance: Focus on Current Controversies

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