A new facile synthetic route to [11C]GSK189254, a selective PET radioligand for imaging of CNS histamine H3 receptor-Reference-Cited by-同舟云学术

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A new facile synthetic route to [11C]GSK189254, a selective PET radioligand for imaging of CNS histamine H3 receptor

Published:2012-07 Issue:14 Volume:22 Page:4713-4718
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Wang Min,Gao Mingzhang,Steele Brandon L.,Glick-Wilson Barbara E.,Brown-Proctor Clive,Shekhar Anantha,Hutchins Gary D.,Zheng Qi-Huang

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference40 articles.

1. Inverse agonist histamine H3 receptor PET tracers labelled with carbon-11 or fluorine-18

2. Synthesis and Evaluation of Structurally Constrained Quinazolinone Derivatives as Potent and Selective Histamine H3 Receptor Inverse Agonists

3. A rat model of changes in dural mast cells and brain histamine receptor H3 expression following traumatic brain injury

4. Evaluation of the binding characteristics of [18F]fluoroproxyfan in the rat brain for in vivo visualization of histamine H3 receptor

5. Histamine Pharmacology and New CNS Drug Targets

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1. Binding of the Dual-Action Anti-Parkinsonian Drug AG-0029 to Dopamine D₂ and Histamine H₃ Receptors: A PET Study in Healthy Rats;Molecular Pharmaceutics;2022-06-22

2. Pharmacokinetic Modeling of [¹¹C]GSK-189254, PET Tracer Targeting H₃ Receptors, in Rat Brain;Molecular Pharmaceutics;2022-02-16

3. A ring expansion strategy towards diverse azaheterocycles;Nature Chemistry;2021-07-19

4. Synthesis of 3-aryl-3-benzazepines via aryne [1,2] Stevens rearrangement of 1,2,3,4-tetrahydroisoquinolines;Organic Chemistry Frontiers;2018

5. Reactions of nitrogen-containing acetals with aromatic nucleophiles;Russian Chemical Reviews;2017-01-26

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