Identification of pyrrolo[2,1-f][1,2,4]triazine-based inhibitors of Met kinase-Reference-Cited by-同舟云学术

Identification of pyrrolo[2,1-f][1,2,4]triazine-based inhibitors of Met kinase

Published:2008-03 Issue:6 Volume:18 Page:1945-1951
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Schroeder Gretchen M.,Chen Xiao-Tao,Williams David K.,Nirschl David S.,Cai Zhen-Wei,Wei Donna,Tokarski John S.,An Yongmi,Sack John,Chen Zhong,Huynh Tram,Vaccaro Wayne,Poss Michael,Wautlet Barri,Gullo-Brown Johnni,Kellar Kristen,Manne Veeraswamy,Hunt John T.,Wong Tai W.,Lombardo Louis J.,Fargnoli Joseph,Borzilleri Robert M.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference29 articles.

1. Discovery of 5-[5-Fluoro-2-oxo-1,2- dihydroindol-(3Z)-ylidenemethyl]-2,4- dimethyl-1H-pyrrole-3-carboxylic Acid (2-Diethylaminoethyl)amide, a Novel Tyrosine Kinase Inhibitor Targeting Vascular Endothelial and Platelet-Derived Growth Factor Receptor Tyrosine Kinase

2. Discovery of N-(2-Chloro-6-methyl- phenyl)-2-(6-(4-(2-hydroxyethyl)- piperazin-1-yl)-2-methylpyrimidin-4- ylamino)thiazole-5-carboxamide (BMS-354825), a Dual Src/Abl Kinase Inhibitor with Potent Antitumor Activity in Preclinical Assays

3. Tyrosine kinase inhibitors in cancer therapy

4. Cancer metastasis therapeutic targets and drug discovery: emerging small-molecule protein kinase inhibitors

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1. Novel 3-phenylquinazolin-2,4(1H,3H)-diones as dual VEGFR-2/c-Met-TK inhibitors: design, synthesis, and biological evaluation;Scientific Reports;2023-10-30

2. Regio- and Diastereoselective 1,3-Dipolar Cycloadditions of 1,2,4-Triazin-1-ium Ylides: a Straightforward Synthetic Route to Polysubstituted Pyrrolo[2,1-f][1,2,4]triazines;ACS Omega;2022-06-10

3. Bicyclic 5-6 Systems With One Bridgehead (Ring Junction) Nitrogen Atom: Two Extra Heteroatoms 0:2;Comprehensive Heterocyclic Chemistry IV;2022

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5. Pyrrolo[2,1-f][1,2,4]triazine: a promising fused heterocycle to target kinases in cancer therapy;Medicinal Chemistry Research;2021-11-13