Fluorinated pyrazole acids are agonists of the high affinity niacin receptor GPR109a-Reference-Cited by-同舟云学术

Fluorinated pyrazole acids are agonists of the high affinity niacin receptor GPR109a

Published:2007-10 Issue:20 Volume:17 Page:5620-5623
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Skinner Philip J.,Cherrier Martin C.,Webb Peter J.,Shin Young-Jun,Gharbaoui Tawfik,Lindstrom Andrew,Hong Vu,Tamura Susan Y.,Dang Huong T.,Pride Cameron C.,Chen Ruoping,Richman Jeremy G.,Connolly Daniel T.,Semple Graeme

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference21 articles.

1. Influence of nicotinic acid on serum cholesterol in man

2. The benefits of niacin in atherosclerosis

3. Nicotinic acid: the broad-spectrum lipid drug. A 50th anniversary review

4. Characterization of a G Protein-Coupled Receptor for Nicotinic Acid

5. The nicotinic acid receptor GPR109A (HM74A or PUMA-G) as a new therapeutic target

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